PDB code | Main view | Title | 1aj6 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1aj6&file=traces.jpg) | NOVOBIOCIN-RESISTANT MUTANT (R136H) OF THE N-TERMINAL 24 KDA FRAGMENT OF DNA GYRASE B COMPLEXED WITH NOVOBIOCIN AT 2.3 ANGSTROMS RESOLUTION |
1bgw | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1bgw&file=traces.jpg) | TOPOISOMERASE RESIDUES 410-1202, |
1bjt | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1bjt&file=traces.jpg) | TOPOISOMERASE II RESIDUES 409-1201 |
1ei1 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1ei1&file=traces.jpg) | DIMERIZATION OF E. COLI DNA GYRASE B PROVIDES A STRUCTURAL MECHANISM FOR ACTIVATING THE ATPASE CATALYTIC CENTER |
1kij | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1kij&file=traces.jpg) | Crystal structure of the 43K ATPase domain of Thermus thermophilus gyrase B in complex with novobiocin |
1kzn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1kzn&file=traces.jpg) | Crystal Structure of E. coli 24kDa Domain in Complex with Clorobiocin |
1pvg | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1pvg&file=traces.jpg) | Crystal Structure of the ATPase region of Saccharomyces Cerevisiae topoisomerase II |
1qzr | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1qzr&file=traces.jpg) | CRYSTAL STRUCTURE OF THE ATPASE REGION OF SACCHAROMYCES CEREVISIAE TOPOISOMERASE II BOUND TO ICRF-187 (DEXRAZOXANE) |
1s14 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1s14&file=traces.jpg) | Crystal structure of Escherichia coli Topoisomerase IV ParE 24kDa subunit |
1s16 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1s16&file=traces.jpg) | Crystal Structure of E. coli Topoisomerase IV ParE 43kDa subunit complexed with ADPNP |
1zxm | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1zxm&file=traces.jpg) | Human Topo IIa ATPase/AMP-PNP |
1zxn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=1zxn&file=traces.jpg) | Human DNA topoisomerase IIa ATPase/ADP |
2rgr | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2rgr&file=traces.jpg) | Topoisomerase IIA bound to G-segment DNA |
2xco | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xco&file=traces.jpg) | The 3.1A crystal structure of the catalytic core (B'A' region) of Staphylococcus aureus DNA Gyrase |
2xcq | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xcq&file=traces.jpg) | The 2.98A crystal structure of the catalytic core (B'A' region) of Staphylococcus aureus DNA Gyrase |
2xcr | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xcr&file=traces.jpg) | The 3.5A crystal structure of the catalytic core (B'A' region) of Staphylococcus aureus DNA Gyrase complexed with GSK299423 and DNA |
2xcs | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xcs&file=traces.jpg) | The 2.1A crystal structure of S. aureus Gyrase complex with GSK299423 and DNA |
2xct | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xct&file=traces.jpg) | The twinned 3.35A structure of S. aureus Gyrase complex with Ciprofloxacin and DNA |
2xkj | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xkj&file=traces.jpg) | CRYSTAL STRUCTURE OF CATALYTIC CORE OF A. BAUMANNII TOPO IV (PARE- PARC FUSION TRUNCATE) |
2xkk | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2xkk&file=traces.jpg) | CRYSTAL STRUCTURE OF MOXIFLOXACIN, DNA, and A. BAUMANNII TOPO IV ( PARE-PARC FUSION TRUNCATE) |
2zjt | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=2zjt&file=traces.jpg) | Crystal structure of dna gyrase B' domain sheds lights on the mechanism for T-segment navigation |
3cwv | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3cwv&file=traces.jpg) | Crystal structure of B-subunit of the DNA gyrase from Myxococcus xanthus |
3foe | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3foe&file=traces.jpg) | Structural insight into the quinolone-DNA cleavage complex of type IIA topoisomerases |
3fof | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3fof&file=traces.jpg) | Structural insight into the quinolone-DNA cleavage complex of type IIA topoisomerases |
3fv5 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3fv5&file=traces.jpg) | Crystal Structure of E. coli Topoisomerase IV co-complexed with inhibitor |
3g75 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3g75&file=traces.jpg) | Crystal structure of Staphylococcus aureus Gyrase B co-complexed with 4-METHYL-5-[3-(METHYLSULFANYL)-1H-PYRAZOL-5-YL]-2-THIOPHEN-2-YL-1,3-THIAZOLE inhibitor |
3g7b | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3g7b&file=traces.jpg) | Staphylococcus aureus Gyrase B co-complex with METHYL ({5-[4-(4-HYDROXYPIPERIDIN-1-YL)-2-PHENYL-1,3-THIAZOL-5-YL]-1H-PYRAZOL-3-YL}METHYL)CARBAMATE inhibitor |
3g7e | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3g7e&file=traces.jpg) | Crystal structure of E. coli Gyrase B co-complexed with PROP-2-YN-1-YL {[5-(4-PIPERIDIN-1-YL-2-PYRIDIN-3-YL-1,3-THIAZOL-5-YL)-1H-PYRAZOL-3-YL]METHYL}CARBAMATE inhibitor |
3ig0 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3ig0&file=traces.jpg) | crystal structure of the second part of the Mycobacterium tuberculosis DNA gyrase reaction core: the TOPRIM domain at 2.1 A resolution |
3k9f | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3k9f&file=traces.jpg) | Detailed structural insight into the quinolone-DNA cleavage complex of type IIA topoisomerases |
3ksa | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3ksa&file=traces.jpg) | Detailed structural insight into the DNA cleavage complex of type IIA topoisomerases (cleaved form) |
3ksb | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3ksb&file=traces.jpg) | Detailed structural insight into the DNA cleavage complex of type IIA topoisomerases (re-sealed form) |
3l4j | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3l4j&file=traces.jpg) | Topoisomerase II-DNA cleavage complex, apo |
3l4k | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3l4k&file=traces.jpg) | Topoisomerase II-DNA cleavage complex, metal-bound |
3lnu | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3lnu&file=traces.jpg) | Crystal structure of ParE subunit |
3lps | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3lps&file=traces.jpg) | Crystal structure of parE |
3ltn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3ltn&file=traces.jpg) | Inhibitor-stabilized topoisomerase IV-DNA cleavage complex (S. pneumoniae) |
3m4i | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3m4i&file=traces.jpg) | Crystal structure of the second part of the Mycobacterium tuberculosis DNA gyrase reaction core: the TOPRIM domain at 1.95 A resolution |
3nuh | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3nuh&file=traces.jpg) | A domain insertion in E. coli GyrB adopts a novel fold that plays a critical role in gyrase function |
3qx3 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3qx3&file=traces.jpg) | Human topoisomerase IIbeta in complex with DNA and etoposide |
3rad | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3rad&file=traces.jpg) | Quinolone(Clinafloxacin)-DNA cleavage complex of type IV topoisomerase from S. pneumoniae |
3rae | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3rae&file=traces.jpg) | Quinolone(Levofloxacin)-DNA cleavage complex of type IV topoisomerase from S. pneumoniae |
3raf | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3raf&file=traces.jpg) | Quinazolinedione-DNA cleavage complex of type IV topoisomerase from S. pneumoniae |
3ttz | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3ttz&file=traces.jpg) | Crystal structure of a topoisomerase ATPase inhibitor |
3u2d | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3u2d&file=traces.jpg) | S. aureus GyrB ATPase domain in complex with small molecule inhibitor |
3u2k | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3u2k&file=traces.jpg) | S. aureus GyrB ATPase domain in complex with a small molecule inhibitor |
3zkb | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3zkb&file=traces.jpg) | CRYSTAL STRUCTURE OF THE ATPASE REGION OF Mycobacterium tuberculosis GyrB WITH AMPPNP |
3zkd | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3zkd&file=traces.jpg) | CRYSTAL STRUCTURE OF THE ATPASE REGION OF Mycobacterium tuberculosis GyrB WITH AMPPNP |
3zm7 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=3zm7&file=traces.jpg) | CRYSTAL STRUCTURE OF THE ATPASE REGION OF Mycobacterium tuberculosis GyrB WITH AMPPCP |
4b6c | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4b6c&file=traces.jpg) | Structure of the M. smegmatis GyrB ATPase domain in complex with an aminopyrazinamide |
4bae | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4bae&file=traces.jpg) | Optimisation of pyrroleamides as mycobacterial GyrB ATPase inhibitors: Structure Activity Relationship and in vivo efficacy in the mouse model of tuberculosis |
4bul | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4bul&file=traces.jpg) | Novel hydroxyl tricyclics (e.g. GSK966587) as potent inhibitors of bacterial type IIA topoisomerases |
4duh | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4duh&file=traces.jpg) | Crystal structure of 24 kDa domain of E. coli DNA gyrase B in complex with small molecule inhibitor |
4em7 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4em7&file=traces.jpg) | Crystal structure of a topoisomerase ATP inhibitor |
4emv | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4emv&file=traces.jpg) | Crystal structure of a topoisomerase ATP inhibitor |
4fm9 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4fm9&file=traces.jpg) | Human topoisomerase II alpha bound to DNA |
4g0u | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4g0u&file=traces.jpg) | Human topoisomerase IIbeta in complex with DNA and amsacrine |
4g0v | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4g0v&file=traces.jpg) | Human topoisomerase iibeta in complex with DNA and mitoxantrone |
4g0w | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4g0w&file=traces.jpg) | Human topoisomerase iibeta in complex with DNA and ametantrone |
4gee | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4gee&file=traces.jpg) | Pyrrolopyrimidine inhibitors of DNA gyrase B and topoisomerase IV, part I: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4gfh | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4gfh&file=traces.jpg) | Topoisomerase II-DNA-AMPPNP complex |
4gfn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4gfn&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic |
4ggl | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4ggl&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity |
4hxw | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hxw&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4hxz | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hxz&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4hy1 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hy1&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4hym | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hym&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4hyp | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hyp&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4hz0 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hz0&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity. |
4hz5 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4hz5&file=traces.jpg) | Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity |
4i3h | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4i3h&file=traces.jpg) | A three-gate structure of topoisomerase IV from Streptococcus pneumoniae |
4j3n | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4j3n&file=traces.jpg) | Human Topoisomerase Iibeta in complex with DNA |
4juo | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4juo&file=traces.jpg) | A low-resolution three-gate structure of topoisomerase IV from Streptococcus pneumoniae in space group H32 |
4k4o | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4k4o&file=traces.jpg) | The DNA Gyrase B ATP binding domain of Enterococcus faecalis in complex with a small molecule inhibitor |
4kfg | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4kfg&file=traces.jpg) | The DNA Gyrase B ATP binding domain of Escherichia coli in complex with a small molecule inhibitor. |
4koe | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4koe&file=traces.jpg) | 4KOE |
4kpe | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4kpe&file=traces.jpg) | 4KPE |
4kpf | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4kpf&file=traces.jpg) | 4KPF |
4kqv | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4kqv&file=traces.jpg) | Topoisomerase iv atp binding domain of francisella tularensis in complex with a small molecule inhibitor |
4ksg | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4ksg&file=traces.jpg) | Dna gyrase atp binding domain of enterococcus faecalis in complex with a small molecule inhibitor (4-[(1S,5R,6R)-6-AMINO-1-METHYL-3-AZABICYCLO[3.2.0]HEPT-3-YL]-6-FLUORO-N-METHYL-2-[(2-METHYLPYRIMIDIN-5-YL)OXY]-9H-PYRIMIDO[4,5-B]INDOL-8-AMINE) |
4ksh | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4ksh&file=traces.jpg) | Dna gyrase atp binding domain of enterococcus faecalis in complex with a small molecule inhibitor (7-({4-[(3R)-3-AMINOPYRROLIDIN-1-YL]-5-CHLORO-6-ETHYL-7H-PYRROLO[2,3-D]PYRIMIDIN-2-YL}SULFANYL)-1,5-NAPHTHYRIDIN-1(4H)-OL) |
4ktn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4ktn&file=traces.jpg) | Dna gyrase atp binding domain of enterococcus faecalis in complex with a small molecule inhibitor ((3S)-1-[2-(PYRIDO[2,3-B]PYRAZIN-7-YLSULFANYL)-9H-PYRIMIDO[4,5-B]INDOL-4-YL]PYRROLIDIN-3-AMINE) |
4lp0 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4lp0&file=traces.jpg) | Crystal structure of a topoisomerase ATP inhibitor |
4lpb | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4lpb&file=traces.jpg) | Crystal structure of a topoisomerase ATPase inhibitor |
4mb9 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4mb9&file=traces.jpg) | Structure of Streptococcus pneumonia ParE in complex with AZ13102335 |
4mbc | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4mbc&file=traces.jpg) | Structure of Streptococcus pneumonia ParE in complex with AZ13053807 |
4mot | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4mot&file=traces.jpg) | Structure of Streptococcus pneumonia pare in complex with AZ13072886 |
4p8o | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4p8o&file=traces.jpg) | 4P8O |
4plb | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4plb&file=traces.jpg) | 4PLB |
4prv | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4prv&file=traces.jpg) | 4PRV |
4prx | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4prx&file=traces.jpg) | 4PRX |
4pu9 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4pu9&file=traces.jpg) | 4PU9 |
4r1f | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4r1f&file=traces.jpg) | 4R1F |
4tma | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4tma&file=traces.jpg) | 4TMA |
4url | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4url&file=traces.jpg) | 4URL |
4urm | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4urm&file=traces.jpg) | 4URM |
4urn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4urn&file=traces.jpg) | 4URN |
4uro | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4uro&file=traces.jpg) | 4URO |
4wub | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4wub&file=traces.jpg) | 4WUB |
4wuc | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4wuc&file=traces.jpg) | 4WUC |
4wud | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4wud&file=traces.jpg) | 4WUD |
4xtj | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4xtj&file=traces.jpg) | 4XTJ |
4z2c | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4z2c&file=traces.jpg) | 4Z2C |
4z2d | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4z2d&file=traces.jpg) | 4Z2D |
4z2e | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4z2e&file=traces.jpg) | 4Z2E |
4z3o | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4z3o&file=traces.jpg) | 4Z3O |
4z4q | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4z4q&file=traces.jpg) | 4Z4Q |
4z53 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4z53&file=traces.jpg) | 4Z53 |
4zvi | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=4zvi&file=traces.jpg) | 4ZVI |
5boc | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5boc&file=traces.jpg) | 5BOC |
5bod | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5bod&file=traces.jpg) | 5BOD |
5bs3 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5bs3&file=traces.jpg) | 5BS3 |
5bs8 | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5bs8&file=traces.jpg) | 5BS8 |
5bta | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5bta&file=traces.jpg) | 5BTA |
5btc | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5btc&file=traces.jpg) | 5BTC |
5btd | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5btd&file=traces.jpg) | 5BTD |
5btf | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5btf&file=traces.jpg) | 5BTF |
5btg | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5btg&file=traces.jpg) | 5BTG |
5bti | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5bti&file=traces.jpg) | 5BTI |
5btl | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5btl&file=traces.jpg) | 5BTL |
5btn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5btn&file=traces.jpg) | 5BTN |
5cdm | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cdm&file=traces.jpg) | 5CDM |
5cdn | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cdn&file=traces.jpg) | 5CDN |
5cdo | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cdo&file=traces.jpg) | 5CDO |
5cdp | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cdp&file=traces.jpg) | 5CDP |
5cdq | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cdq&file=traces.jpg) | 5CDQ |
5cdr | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cdr&file=traces.jpg) | 5CDR |
5cph | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cph&file=traces.jpg) | 5CPH |
5ctu | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5ctu&file=traces.jpg) | 5CTU |
5ctw | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5ctw&file=traces.jpg) | 5CTW |
5ctx | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5ctx&file=traces.jpg) | 5CTX |
5cty | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5cty&file=traces.jpg) | 5CTY |
5d6p | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5d6p&file=traces.jpg) | 5D6P |
5d6q | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5d6q&file=traces.jpg) | 5D6Q |
5d7c | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5d7c&file=traces.jpg) | 5D7C |
5d7d | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5d7d&file=traces.jpg) | 5D7D |
5d7r | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5d7r&file=traces.jpg) | 5D7R |
5eix | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5eix&file=traces.jpg) | 5EIX |
5iwi | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5iwi&file=traces.jpg) | 5IWI |
5iwm | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5iwm&file=traces.jpg) | 5IWM |
5l3j | ![](http://www.ebi.ac.uk/thornton-srv/databases/cgi-bin/pdbsum/getimg.pl?source=pdbsum&pdb_code=5l3j&file=traces.jpg) | 5L3J |